Actifast

Actifast Uses, Dosage, Side Effects, Mechanism of Action, How Long Does it Take to Work? Actifast is a brand name. Its generic name is Ketorolac.

Actifast

Actifast, also known as toradol, is a non-steroidal anti-inflammatory drug (NSAID) used to treat pain and inflammation. It is available without a prescription for the relief of mild to moderate pain, but may be administered in a hospital for more severe pain.

Uses for

Actifast is used to relieve moderate to severe pain, including pain after surgery and pain from injuries. It can be used to treat pain associated with sprains, strains, tendonitis, myositis, bursitis, discitis, periodontal abscess, and dental surgery. It is also used to reduce fever and pain associated with osteoarthritis and rheumatoid arthritis.

Mechanism of Action

Actifast works by reducing hormones that cause pain and inflammation in the body. It stops the production of prostaglandins, which are compounds in the body that can cause pain, inflammation, and fever. By inhibiting the formation of these compounds, ketorolac can reduce pain and inflammation.

How long does it take to work?

Actifast usually begins to work within 30 minutes of taking it. The effects of the medication can last up to 6 hours.

Absorption

Actifast is rapidly and completely absorbed from the gastrointestinal tract. It has an absolute bioavailability of approximately 70%.

Route of Elimination

Actifast is eliminated mainly through the kidneys as metabolites or unchanged drug. It is also excreted in small amounts in the bile.

Dosage

The recommended dose of Actifast is 10-60 mg every 4-6 hours, with a maximum dose of 120 mg per day. The maximum duration of treatment is 5 days.

Administration

Actifast can be taken orally or administered intravenously. It is usually taken with food or milk to minimize the risk of stomach upset.

Side Effects

Some common side effects of ketorolac may include headache, dizziness, nausea, vomiting, stomach upset, heartburn, and increased risk of bleeding or stomach ulcers. Less common side effects may include dizziness, rash, and unusual bleeding or bruising.

Toxicity

Actifast is generally safe and well tolerated when taken as directed. However, taking high doses or using for long periods of time can increase the risk of side effects, including kidney damage, gastrointestinal bleeding, and stomach ulcers. Overdose can occur if more than the recommended dose is taken.

Precautions

Patients should tell their doctor or healthcare provider if they have had any type of surgery, kidney or liver disease, asthma, heart disease, bleeding disorders, or any other medical conditions before taking ketorolac. It is important to tell the doctor or healthcare provider about all the medicines taken, including prescription and nonprescription medicines, vitamins, and herbal supplements.

Interactions

Actifast can interact with other medications, including other anti-inflammatory drugs, anticoagulants, lithium, methotrexate, and other NSAIDs. Patients should tell their doctor or healthcare provider about all the medicines taken in order to avoid any potential drug interactions.

Disease Interactions

Actifast may interact with certain diseases, including kidney or liver disease, asthma, recent surgery, bleeding disorders, heart disease, and other medical conditions. Patients should tell their doctor or healthcare provider about any medical conditions before taking ketorolac.

Drug Interactions

Actifast can interact with other medications, including other NSAIDs, anticoagulants, lithium, methotrexate, and other prescription and non-prescription medications. Patients should tell their doctor or healthcare provider about all the medicines taken in order to avoid any potential drug interactions.

Food Interactions

Actifast should be taken with food or milk to reduce the risk of stomach upset. It is important to tell the doctor or healthcare provider about any dietary supplements or vitamins taken in order to avoid any potential food interactions.

Pregnancy Use

Actifast should not be used by pregnant women, unless specifically recommended by a doctor. Use of this medication during the third trimester of pregnancy may cause side effects in the baby. Patients should tell their doctor or healthcare provider if they are pregnant before starting this medication.

Lactation Use

Actifast should not be used while breastfeeding, unless specifically recommended by a doctor. Patients should tell their doctor or healthcare provider if they are breastfeeding before starting this medication.

Acute Overdose

Acute overdose of ketorolac can cause excessive sedation, hypotension, shock, coma, and death. If significant amounts have been ingested, contact a poison control center for advice.

Contraindication

Actifast should not be used in patients with active peptic ulcer, bleeding problems, kidney or liver dysfunction, known hypersensitivity or allergy to this medication, or in patients who are taking other medications that interact with ketorolac.

Use Direction

Actifast comes in tablet or intravenous form and is to be taken or administered according to directions provided by a doctor or healthcare provider. Patients should tell their doctor or healthcare provider if they are pregnant or breastfeeding before starting this medication.

Storage Condition

Actifast should be stored in a cool, dry place, away from light and moisture. Keep all medication out of the reach of children.

Volume of Distribution

Actifast has a volume of distribution of 0.6-1.2 L/kg.

Half Life

Actifast has a half-life of 4-6 hours.

Clearance

Actifast has a clearance of 2-4 L/h.

Here you find in details version of Actifast

Some Frequently Asked Questions About Actifast

What is Actifast?

Actifast is a nonsteroidal anti-inflammatory drug (NSAID) used to treat pain and inflammation. It is sold under the brand names Toradol, Acular LS, Cashol, and Acupain, as well as generic forms.

How does Actifast work?

Actifast works by blocking the production of hormones that cause inflammation and pain in the body. This helps to reduce pain and swelling.

What are the side effects of Actifast?

The most common side effects of ketorolac include stomach upset, nausea, vomiting, and diarrhea. Other side effects may include headaches, dizziness, rashes, and fluid retention.

Should I take Actifast with food or on an empty stomach?

It is recommended to take ketorolac with food, as this may help reduce the risk of stomach upset.

What should I do if I experience side effects from taking Actifast?

If you experience any side effects while taking ketorolac, you should contact your doctor for advice. Depending on the severity, your doctor may recommend that you stop taking ketorolac.

Can I take Actifast with other medications?

You should always check with your doctor before taking any medication, including ketorolac, with other medications. Some medications may interact with ketorolac and increase the risk of side effects or reduce its effectiveness.

What is the recommended dosage of Actifast?

The recommended dosage of ketorolac depends on your medical condition and the brand or generic form you are taking. Your doctor will advise you on the correct dosage.

Can I take Actifast if I am pregnant?

No. Actifast should not be taken if you are pregnant unless specifically advised by your doctor.

Can I take Actifast if I am breastfeeding?

No. Actifast should not be taken if you are breastfeeding unless specifically advised by your doctor.

Are there any people who should not take Actifast?

Actifast should not be taken by people who are allergic to nonsteroidal anti-inflammatory drugs (NSAIDs) or by those who have had asthma, hives, or other allergic reactions caused by NSAIDs. People who have had a history of stomach or intestinal bleeding or ulcers should also avoid taking ketorolac.

Can I take Actifast if I have high blood pressure?

Yes, you can take ketorolac if you have high blood pressure. However, you should be monitored closely for potential changes in your blood pressure while taking this medication.

What does Actifast treat?

Actifast is used to treat pain and inflammation caused by a variety of conditions including arthritis, tendinitis, bursitis, and menstrual cramps.

How long does it take for Actifast to take effect?

The effects of ketorolac can be seen within an hour of taking the medication. However, it may take time for the full therapeutic effects of the medication to be seen.

How long do the effects of Actifast last?

Most people will experience relief from ketorolac for up to six hours, depending on the dose and the condition being treated.

Should I take more than the recommended dose of Actifast?

No. You should not take more than the recommended dose of ketorolac as this can increase the risk of serious side effects.

Can I take Actifast with acetaminophen?

No. You should not take acetaminophen with ketorolac as this can increase the risk of serious side effects.

Can I take Actifast with ibuprofen?

No. You should not take ibuprofen with ketorolac as this can increase the risk of serious side effects.

Can I drink alcohol while taking Actifast?

No. You should not drink alcohol while taking ketorolac as this can increase the risk of serious side effects.

Can I take Actifast with birth control?

Yes. It is generally safe to take ketorolac with birth control, although you should always check with your doctor to be sure.

Are there any supplements I should avoid while on Actifast?

Yes. You should avoid taking supplements containing St. John's Wort while taking ketorolac, as this can increase the risk of serious side effects and may reduce the effectiveness of the medication.

Can I take Actifast if I have a history of ulcers?

No. If you have a history of ulcers, you should not take ketorolac as this can increase the risk of serious side effects.